Saussurea lappa

Ethnobotanical Studies

Studies

High throughput virtual screening and validation of Plant-Based EGFR L858R kinase inhibitors against Non-Small cell lung Cancer: An integrated approach Utilizing GC-MS, network Pharmacology, Docking, and molecular dynamics.

Summary

Researchers identified potential inhibitors from Dehydrocostus lactone and Mokkolactone for EGFR L858R mutant lung cancer. These compounds showed anti-proliferative activity and stable binding in molecular simulations. Further in vivo studies are needed for efficacy assessment.

Gao K et al (2024).
Saudi Pharm J.
PubMed:
39139718

Comparative Efficacy of Aristolochia rotunda L. (Zarawand Mudaharaj) and Saussurea lappa C.B. Clarke (Qust) in Primary Dysmenorrhea--A Single-Blind Randomized Clinical Study.

Sumaiya S et al (2024).
Altern Ther Health Med.
PubMed:
39110054

From nature's bounty to drug discovery: Leveraging phytochemicals and molecular approaches to combat multi-drug-resistant (MDR) tuberculosis.

Review
Nalam SM et al (2024).
Indian J Tuberc.
PubMed:
39067943

Lappanolides A-N, fourteen undescribed sesquiterpenoids from Saussurea costus (Syn. Saussurea lappa) and their anti HBV activity.

Li HB et al (2024).
Phytochemistry.
PubMed:
38972443

The effect of dietary administration of Saussurea lappa root on performance, blood biochemical indices, redox status, innate immune response, intestinal microbial population and resistance against A. hydrophila infections of Tilapia Fingerlings.

Naiel MAE et al (2024).
J Anim Physiol Anim Nutr (Berl).
PubMed:
38851860

A sustainable approach to prepare green synthesis of copper nanoparticles of Bauhinia variegata & Saussurea lappa: Unveiling in-vitro anti-obesity applications.

Summary

Flower extracts were used to synthesize copper nanoparticles with potential applications in stabilizing compounds, antimicrobial activity, and anti-obesity/anti-diabetic effects. This study demonstrates the versatility and benefits of using plant-synthesized nanoparticles in various fields.

Kumar M et al (2024).
Heliyon.
PubMed:
38644870

Impact of Saussurea lappa against foodborne parasite Trichinella spiralis experimental infections induced variation in DNA damage, oxidative stress and PCNA expression in rat skeletal muscles.

Alghabban AJM et al (2024).
Toxicol Res (Camb).
PubMed:
38529200

Dehydrocostus lactone suppresses gastric cancer progression by targeting ACLY to inhibit fatty acid synthesis and autophagic flux.

Summary

Dehy, a compound from Saussurea lappa Clarke, effectively treats cancer and gastrointestinal disorders. However, its specific impact on gastric cancer is not well-known.

Chen Y et al (2024).
J Adv Res.
PubMed:
38295877

Optimized bilosome-based nanoparticles enhance cytotoxic and pro-apoptotic activity of costunolide in LS174T colon cancer cells.

Summary

Researchers developed a nanoformulation of costunolide (COST) to improve its anti-proliferative effects in colon cancer cells. The optimized formulation showed increased cytotoxicity, enhanced apoptosis, and altered gene expression compared to raw COST, making it more effective in killing cancer cells.

Alamoudi AJ et al (2023).
Biomed Pharmacother.
PubMed:
37897972

Costunolide alleviated DDC induced ductular reaction and inflammatory response in murine model of cholestatic liver disease.

Hao J et al (2023).
J Tradit Complement Med.
PubMed:
37396159

Secondary Metabolites Generated from Saussurea lappa and Ligusticum sinensis Essential Oils by Microwave-Assisted Hydrodistillation: in-silico Molecular Docking and in-vitro Antibacterial Efficacy.

Hegazy ME et al (2023).
Chem Biodivers.
PubMed:
37358062

Undescribed amino acid-sesquiterpene lactone adducts and sesquiterpene glycosides from the roots of Saussurea lappa and their anti-HBV activity.

Cong XY et al (2023).
Fitoterapia.
PubMed:
37321417

Investigation of the antiviral effects of Saussurea lappa root extract against SARS-CoV-2 virus.

Summary

Researchers found that a plant extract from Saussurea lappa roots could potentially be used as a food supplement to combat SARS-CoV-2, as it showed some ability to inhibit the virus. Further research is needed to establish its effectiveness as a treatment for COVID-19.

Polat HU et al (2023).
Mol Nutr Food Res.
PubMed:
37170075

Integrated analysis of smRNAome, transcriptome, and degradome data to decipher microRNAs regulating costunolide biosynthesis in Saussurea lappa.

Kaur R et al (2023).
Plant Sci.
PubMed:
36965630

Costunolide covalently targets NACHT domain of NLRP3 to inhibit inflammasome activation and alleviate NLRP3-driven inflammatory diseases.

Xu H et al (2023).
Acta Pharm Sin B.
PubMed:
36873170

Investigation of Molecular Mechanisms Involved in Sensitivity to the Anti-Cancer Activity of Costunolide in Breast Cancer Cells.

Choi YJ et al (2023).
Int J Mol Sci.
PubMed:
36835418

Impact of Saussurea lappa root extract against copper oxide nanoparticles induced oxidative stress and toxicity in rat cardiac tissues.

Tousson E and El-Gharbawy DM (2023).
Environ Toxicol.
PubMed:
36286243

Emergence of high colistin resistance in carbapenem resistant Acinetobacter baumannii in Pakistan and its potential management through immunomodulatory effect of an extract from Saussurea lappa.

Ahsan U et al (2022).
Front Pharmacol.
PubMed:
36188613

Protective and therapeutic potentials of HDL and ApoA1 in COVID-19 elderly and chronic illness patients.

Summary

Scientists have discovered that HDL, a protein responsible for various functions in the body, is affected by alterations in its structure caused by SARS-CoV-2. This discovery sheds light on the increased risk of severe COVID-19 in older adults, obese individuals, and those with chronic illnesses. The study's findings could potentially lead to new treatments that target HDL to improve outcomes for these vulnerable populations.

Review COVID-19
AbdelHafez MA et al (2022).
Bull Natl Res Cent.
PubMed:
35915785

The exploration of bio-inspired copper oxide nanoparticles: synthesis, characterization and in-vitro biological investigations.

Kolahalam LA et al (2022).
Heliyon.
PubMed:
35770152

Tentatively Identified (UPLC/T-TOF-MS/MS) Compounds in the Extract of Saussurea costus Roots Exhibit In Vivo Hepatoprotection via Modulation of HNF-1α, Sirtuin-1, C/ebpα, miRNA-34a and miRNA-223.

El Gizawy HA et al (2022).
Molecules.
PubMed:
35566153

Structure-Based Molecular Networking for the Discovery of Anti-HBV Compounds from Saussurea lappa (Decne.) C.B Clarke.

Wu T et al (2022).
Molecules.
PubMed:
35335386

Deciphering chemical profiling, pharmacological responses and potential bioactive constituents of Saussurea lappa Decne. Extracts through in vitro approaches.

Naseer S et al (2022).
Saudi J Biol Sci.
PubMed:
35280548

Inhibition of thioredoxin-interacting protein may enhance the therapeutic effect of dehydrocostus lactone in cardiomyocytes under doxorubicin stimulation via the inhibition of the inflammatory response.

Zhang X, Chu C and Huang Y (2022).
Exp Ther Med.
PubMed:
35222703

Curcumae Longae Rhizoma and Saussureae Radix Inhibit Nitric Oxide Production and Cannabinoid Receptor 2 Down-regulation.

Tanikawa T et al (2022).
In Vivo.
PubMed:
34972719